Drugs: Exam 2

Antacids

Aluminum hydroxide, magnesium hydroxide, calcium carbonate

H2 receptor blockers

Cimetidine, famotidine, ranitidine, nizatidine

Proton pump inhibitors

Omeprazole, esomeprazole

Mucosal protective agents

Sucralfate, bismuth subsalicylate, misoprostol

Antimuscarinics

Pirenzepine, dicyclomine

Antimicrobials

Clarithromycin, amoxicillin, metronidazole, tetracycline

Prokinetic drugs

Metoclopramide, cisapride

Laxatives

Senna, bisacodyl, castor oil, methylcellulose, psyllium, bran, magnesium salts, magnesium hydroxide, lactulose, polyethylene glycol, docusate, mineral oil, glycerine

Antiemetics

Antimuscarinic: scopolamine
H1 receptor antagonists: dimehydramine, dimenhydrinate, meclizine, cyclizine
5HT3 receptor blockers: ondansetron, granisetron
D2 antagonists: prochlorperazine, droperidol, haloperidol
Benzodiazepines: lorazepam, alprazolam
Cort

Emetics

Apomorphine, ipecac syrup

Antidiarrheals

Diphenoxylate, loperamide, octreotide, bismuth subsalicylate

Drugs for IBD

Mesalamine, sulfasalazine, infliximab, methotrexate, 6-mercaptopurine, prednisone, prednisolone

Drugs for IBS

Loperamide, diphenoxylate, codeine, hyoscyamine, dicyclomine, alosetron

Pancreatic enzymes

Lipase, alpha-amylase, trypsin, chymotrypsin

NSAIDs

Aspirin, diclofenac, ibuprofen, indomethacin, ketorolac, naproxen, piroxicam, tolmetin, celecoxib, etoricoxib, meloxicam, acetaminophen, acetylcysteine

DMARDs

Methotrexate, cyclophosphamide, azathioprine, leflunomide, hydroxychloroquine, sulfasalazine, gold sodium thiomalate, auranofin, adalimumab, infliximab, etanercept, anakinra, glucocorticoids

Drugs for acute gout

Indomethacin (& other NSAIDs), colchicine, glucocorticoids

Drugs for chronic gout

Allopurinol, probenecid, sulfinpyrazone, rasburicase

Opioid agonists

Morphine, hydromorphone, oxymorphone, heroin, meperidine, fentanyl, sufentanil, alfentanil, remifentanil, methadone, levorphanol, codeine, oxycodone, hydrocodone, propoxyphene, tramadol

Opioid mixed agonist-antagonists

Pentazocine, butorphanol, nalbuphine, buprenorphine

Opioid antagonists

Naloxone, naltrexone

Antitussives

Dextrometorphan, codeine

Antimotility agents

Diphenoxylate, loperamide

Nonopioid analgesics

Acetaminophen, NSAIDs

Analgesic adjunctive agents

Amitriptyline, imipramine, venlafaxine, duloxetine, carbamazepine, gabapentin, pregabalin, valproate, topiramate, dexamethasone, hydroxyzine, clonidine, lidocaine, capsaicin, caffeine

Adjuvants for pain management

Hydroxyzine, diphenhydramine, senna, bisacodyl, docusate, magnesium hydroxide, lactulose, metoclopramide, prochlorperazine, amphetamine, methylphenidate, naloxone

Drugs to treat immediate allergy

Epinephrine, beta-agonists, corticosteroids, H1 receptor antagonists

Penicillins

Classical: penicillin G, penicillin G benzathine, penicillin G procaine, penicillin V
Extended spectrum: amoxicillin, ampicillin
Anti-staph: methicillin, oxacillin, nafcillin, dicloxacillin
Anti-pseudomonal: piperacillin, ticarcillin, carbenicillin

Cephalosporins

1st gen: cefazolin, cephalexin
2nd gen: cefamandole, cefaclor, cefoxitin, cefotetan
3rd gen: cefoperazone, ceftazidime, cefotaxime, ceftriaxone, cefixime
4th gen: cefepime

Carbapenems

Imipenem, meropenem

Dihydropeptidase inhibitor

Cilastatin

Monobactams

Aztreonam

Beta-lactamase inhibitors

Clavulanic acid, sulbactam, tazobactam

Miscellaneous cell wall synthesis inhibitors

Vancomycin, daptomycin, bacitracin, fosfomycin

Tetracyclines

Tetracycline, doxycycline, minocycline

Glycylcyclines

Tigecycline

Aminogycosides

Amikacin, gentamicin, neomycin, netilmycin, streptomycin, tobramycin

Macrolides

Azithromycin, clarithromycin, erythromycin, telithromycin

Streptogramins

Dalfopristin, quinupristin

Miscellaneous protein synthesis inhibitors

Chloramphenicol, clindamycin, linezolid

Quinolones

1st gen: nalidixic acid
2nd gen: ciprofloxacin
3rd gen: levofloxacin
4th gen: moxifloxacin, gemifloxacin

Sulfonamides

Sulfacetamide, sulfadiazine, sulfadoxine, sulfamethoxazole, sulfasalazine, sulfisoxazole

Other nucleic acid synthesis effectors

Trimethoprim, co-trimoxazole, metronidazole, nitrofurantoin

Anti-mycobacterials

Amikacin, levofloxacin, clofazimine, dapsone, ethambutol, ethionamide, isoniazid, pyrazinamide, rifabutin, rifampin, rifapentine, streptomycin, clarithromycin, minocycline, doxycycline, sulfonamides, cefoxitin, imipenem

Neuraminidase inhibitors

Oseltamivir, zanamivir

Anti-viral ion channel blockers

Amantadine, rimantadine

Synthetic guanosine analog

Ribavirin

Interferons

Interferon alpha, beta, gamma

Nucleotide/nucleoside analogs

Adefovir, entecavir, lamivudine, telbivudine

Purine/pyrimidine analogs

Acyclovir, cidofovir, famciclovir, ganciclovir, penciclovir, trifluridine, valcyclovir, vidarabine

Antisense oligonucleotide

Fomivirsen

Phosphonoformate

Foscarnet

NRTIs

Abacavir, didanosine, emtricitabine, lamivudine, stavudine, tenofovir, zidovudine

NNRTIs

Delavirdine, efavirenz, etravirine, nevirapine

Protease inhibitors

Atazanavir, darunavir, fosamprenavir, indinavir, lopinavir, nelfinavir, ritonavir, saquinavir, tipranavir

Fusion inhibitors

Enfuvirtide, maraviroc

Integrase inhibitor

Raltegravir

Polyenes

Amphotericin B, nystatin

Azoles

Ketoconazole, fluconazole, itraconazole, voriconazole, posaconazole, clotrimazole, miconazole

Allylamines

Terbinafine

Pyrimidine analog

Flucytosine

Echinocandins

Caspofungin

Miscellaneous antifungals

Griseofulvin

Drugs for PCP treatment

Co-trimoxazole, clindamycin, primaquine, dapsone, atovaquone, pentamidine, prednisone

Antiamebics

Metronidazole, tinidazole, diloxanide furoate, iodoquinol, paromomycin, chloroquine, dehydroemetine, emetine, tetracycline

Antihelminthics

Albendazole, mebendazole, thiabendazole, bithionol, diethylcarbamazine, doxycycline, ivermectin, niclosamide, piperazine, praziquantel, pyrantel pamoate

Other antiparasitics

Clindamycin, folinic acid, melarsoprol, metronidazole, nifurtimox, pentamidine, pyrimethamine, sodium stibogluconate, sulfadiazine, suramin, co-trimoxazole

Antimalarials

Artemisinins, atovaquone, chloroquine, clindamycine, doxycycline, halofantrine, lumefantrine, mefloquine, primaquine, proguanil, quinidine, quinine, sulfadoxine, pyrimethamine

Antimetabolites

5-fluorouracil, 6-mercaptopurine, 6-thioguanine, capecitabine, cytarabine, gemcitabine, methotrexate

Antitumor antibiotics

Bleomycin, dactinomycin, daunorubicin, doxorubicin

Epipodophyllotoxins

Etoposide, teniposide

Vinca alkaloids

Vincristine, vinblastine, vinrelbine

Taxanes

Docetaxel, paclitaxel

Captothecins

Irinotecan, topotecan

Nitrogen mustards

Chlorambucil, cyclophosphamide, ifosfamide, mechlorethamine, melphalan

Alkyl sulfonates

Busulfan

Nitrosoureas

Carmustine, lomustine, semustine

Triazenes

Dacarbazine

Methylhydrazines

Procarbazine

Platinum compounds

Cisplatin, carboplatin, oxaliplatin

Glucocorticoids

Dexamethasone, hydrocortisone, prednisolone, prednisone

Estrogens

Diethylstilbestrol, ethinylestradiol

Estrogen inhibitors

Aminoglutethemide, anastrozole, exemestane, formestane, letrozole, tamoxifen, raloxifen

Progestins

Hydroxyprogesterone, megestrol

Androgens

Fluoxymesterone, testosterone

Androgen inhibitors

Goserelin, leuprolide

Androgen receptor blockers

Flutamide

Signal transduction inhibitors

Bortezomib, Cetuximab, erlotinib, gefitinib, imatinib, lapatinib, sorafenib, sunitinib, trastuzumab

Miscellaneous anti-cancer drugs/adjuvants

Arsenic trioxide, hydroxyurea, interferon 2-alpha, interferon 2-beta, L-asparaginase, leucovorin, dexrazoxane, filgrastim, mesna, amifostine

T-cell inhibitors

Cyclosporine, tacrolimus, sirolimus

Cytotoxic drugs

Azathioprine, methotrexate, mycophenolate, cyclophosphamide

Glucocorticoids

Prednisone

Polyclonal antibodies

Antithymocite globulin, rho(D) immunoglobulin, hyperimmune immunoglobulins

Monoclonal antibodies

Infliximab, abciximab, muromonab-CD3, rituximab, daclizumab, cetuximab, basiliximab, etanercept

Other immunosuppressants

Thalidomide

Immunostimulant vaccines

BCG

Immunostimulant cytokines

Interferons, aldesleukin