Drugs for Men's Health and Reproductive Disorders

What is the role of Phosphodieterase in men's health?

Secreted to counteract vasodilation

What is the mechanism of action for sexual dysfunction of a male?

cGMP - vasodilation - corpus cavernosum - phosphodieterase

What drugs cause sexual dysfunction in a male?

Antidepressants
Antihistamines
Antihypertensives
Antiulcer
Sedatives and recreational drugs

What physiological disorders affect men's sexual health?

Diabetes mellitus
Coronary artery disease
Vascular disease

Sildenafil citrate

Viagra

Sildenaful citrate onset

30-60 minutes

Sildenaful citrate duration

4 hours

Vardenaful

Levitra

Vardenaful onset

25-30 minutes

Vardenaful duration

4-5 hours

Tadalafil

Cialis

Tadalafil onset

15-60 minutes

Tadalafil duration

24-36 hours

Avanafil

Stendra

Avanafil onset

15-60 minutes

Avanafil duration

24-36 hours

Side effects of men's sexual dysfunction medications

Headache
Dyspnea
Dizziness
Vision changes
Painful/cloudy urination

What is important for the patient to avoid when taking men's sexual dysfunction medication?

No nitrates because it also causes vasodilation leading to hypotension

5-alpha reductase inhibitors

Inhibits an enzyme in the prostate which causes decreased prostate growth

How long does it take for 5-alpha reductase inhibitors to work?

Up to 6 months

Who cannot handle 5-alpha reductase inhibitors?

Pregnant women because there is a risk of absorption through skin that could affect fetus

What cancer does 5 alpha reductase inhibitors increase the risk of developing?

Prostate

Finasteride

Proscar
5-alpha reductase inhibitor

Duastride

Avodart
5-alpha reductase inhibitor

Alpha- adrenergic blocking agents

Causes vasodilation within urethra to open space and vasoconstrictor prostate so man can pass more urine through the urethra

What is a significant risk of Alpha-adrenergic blocking agents?

Hypotension (especially orthostatic hypotension)

What patient education is needed for alpha adrenergic blocking agents?

Slowly sit/stand up
If encountering dizziness/lightheadedness- need to sit down

First dose effect and alpha adrenergic blocking agents

Risk of hypotension, especially after first dose, patient needs to be monitored frequently with BP

What are safety precautions for alpha adrenergic blocking agents?

Use call bell, don't get up without assistance

Tamsulosin

Flomax
Alpha adrenergic blocking agent

Doxazosin

Cardura
Alpha adrenergic blocking agent

Terasozin

Hytrin
Alpha adrenergic blocking agent